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Tricyclic antipsychotics and antidepressants can inhibit α5-containing GABAA receptors by two distinct mechanisms. , Bampali K., Br J Pharmacol. July 1, 2022; 179 (14): 3675-3692.
GABAA Receptor Subunit Composition Drives Its Sensitivity to the Insecticide Fipronil. , Soualah Z., Front Neurosci. January 1, 2021; 15 768466.
Analysis of Modulation of the ρ1 GABAA Receptor by Combinations of Inhibitory and Potentiating Neurosteroids Reveals Shared and Distinct Binding Sites. , Germann AL., Mol Pharmacol. October 1, 2020; 98 (4): 280-291.
Erythropoietin Increases GABAA Currents in Human Cortex from TLE Patients. , Roseti C., Neuroscience. July 15, 2020; 439 153-162.
Cofactor-enabled functional expression of fruit fly, honeybee, and bumblebee nicotinic receptors reveals picomolar neonicotinoid actions. , Ihara M., Proc Natl Acad Sci U S A. July 14, 2020; 117 (28): 16283-16291.
Differential modulation of human GABAC-ρ1 receptor by sulfur-containing compounds structurally related to taurine. , Ochoa-de la Paz LD., BMC Neurosci. August 3, 2018; 19 (1): 47.
Direct intertectal inputs are an integral component of the bilateral sensorimotor circuit for behavior in Xenopus tadpoles. , Gambrill AC., J Neurophysiol. May 1, 2018; 119 (5): 1947-1961.
Mutation of the inhibitory ethanol site in GABAA ρ1 receptors promotes tolerance to ethanol-induced motor incoordination. , Blednov YA., Neuropharmacology. September 1, 2017; 123 201-209.
Assembly rules for GABAA receptor complexes in the brain. , Martenson JS., Elife. August 17, 2017; 6
Novel Molecule Exhibiting Selective Affinity for GABAA Receptor Subtypes. , Borghese CM., Sci Rep. July 24, 2017; 7 (1): 6230.
GABAB receptor attenuation of GABAA currents in neurons of the mammalian central nervous system. , Shen W., Physiol Rep. March 1, 2017; 5 (6):
The Effect of 4-hydroxybenzaldehyde on the γ-aminobutyric Acid Type A Receptor. , Zhang J., Malays J Med Sci. March 1, 2017; 24 (2): 94-99.
Direct activation of GABAA receptors by substances in the organic acid fraction of Japanese sake. , Izu H., Food Chem. January 1, 2017; 214 354-359.
α7-nAChR agonist enhances neural plasticity in the hippocampus via a GABAergic circuit. , Townsend M., J Neurophysiol. December 1, 2016; 116 (6): 2663-2675.
Allosteric binding site in a Cys-loop receptor ligand-binding domain unveiled in the crystal structure of ELIC in complex with chlorpromazine. , Nys M., Proc Natl Acad Sci U S A. October 25, 2016; 113 (43): E6696-E6703.
Fragile X mental retardation protein knockdown in the developing Xenopus tadpole optic tectum results in enhanced feedforward inhibition and behavioral deficits. , Truszkowski TL., Neural Dev. August 8, 2016; 11 (1): 14.
Analysis of β-Subunit-dependent GABAA Receptor Modulation and Behavioral Effects of Valerenic Acid Derivatives. , Khom S., J Pharmacol Exp Ther. June 1, 2016; 357 (3): 580-90.
Pharmacological induction of skin pigmentation unveils the neuroendocrine circuit regulated by light. , Bertolesi GE ., Pigment Cell Melanoma Res. March 1, 2016; 29 (2): 186-98.
Interactions of L-3,5,3'-Triiodothyronine [corrected], Allopregnanolone, and Ivermectin with the GABAA Receptor: Evidence for Overlapping Intersubunit Binding Modes. , Westergard T., PLoS One. September 4, 2015; 10 (9): e0139072.
Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site. , Middendorp SJ., Neuropharmacology. August 1, 2015; 95 459-67.
Inhibitory effects of insulin on GABAA currents modulated by the GABAA alpha subunit. , Williams DB., J Recept Signal Transduct Res. January 1, 2015; 35 (6): 516-22.
Probing α4βδ GABAA receptor heterogeneity: differential regional effects of a functionally selective α4β1δ/α4β3δ receptor agonist on tonic and phasic inhibition in rat brain. , Hoestgaard-Jensen K., J Neurosci. December 3, 2014; 34 (49): 16256-72.
A cycloartane glycoside derived from Actaea racemosa L. modulates GABAA receptors and induces pronounced sedation in mice. , Strommer B., J Pharmacol Exp Ther. November 1, 2014; 351 (2): 234-42.
Efficient modulation of γ-aminobutyric acid type A receptors by piperine derivatives. , Schöffmann A., J Med Chem. July 10, 2014; 57 (13): 5602-19.
Generation of recombinant antibodies to rat GABAA receptor subunits by affinity selection on synthetic peptides. , Koduvayur SP., PLoS One. February 19, 2014; 9 (2): e87964.
Mutations at beta N265 in γ-aminobutyric acid type A receptors alter both binding affinity and efficacy of potent anesthetics. , Stewart DS., PLoS One. January 1, 2014; 9 (10): e111470.
GABAA receptors containing ρ1 subunits contribute to in vivo effects of ethanol in mice. , Blednov YA., PLoS One. January 1, 2014; 9 (1): e85525.
The orthosteric GABAA receptor ligand Thio-4-PIOL displays distinctly different functional properties at synaptic and extrasynaptic receptors. , Hoestgaard-Jensen K., Br J Pharmacol. October 1, 2013; 170 (4): 919-32.
Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α1 GABA(A) receptors. , Joksimović S., Eur Neuropsychopharmacol. May 1, 2013; 23 (5): 390-9.
Partial agonism of taurine at gamma-containing native and recombinant GABAA receptors. , Kletke O., PLoS One. January 1, 2013; 8 (4): e61733.
A single amino acid determines the toxicity of Ginkgo biloba extracts. , Thompson AJ., FASEB J. May 1, 2012; 26 (5): 1884-91.
Modulation of human GABAA receptor function: a novel mode of action of drugs of abuse. , Hondebrink L., Neurotoxicology. December 1, 2011; 32 (6): 823-7.
Cloning and characterization of GABAA α subunits and GABAB subunits in Xenopus laevis during development. , Kaeser GE., Dev Dyn. April 1, 2011; 240 (4): 862-73.
Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site. , Thompson AJ., Neuropharmacology. January 1, 2011; 60 (2-3): 488-95.
GABAergic circuits control stimulus-instructed receptive field development in the optic tectum. , Richards BA., Nat Neurosci. September 1, 2010; 13 (9): 1098-106.
Fragrant dioxane derivatives identify beta1-subunit-containing GABAA receptors. , Sergeeva OA., J Biol Chem. July 30, 2010; 285 (31): 23985-93.
Agonist function of the recombinant alpha 4 beta 3 delta GABAA receptor is dependent on the human and rat variants of the alpha 4-subunit. , Wang MD., Clin Exp Pharmacol Physiol. July 1, 2010; 37 (7): 662-9.
About a snail, a toad, and rodents: animal models for adaptation research. , Roubos EW ., Front Endocrinol (Lausanne). January 1, 2010; 1 4.
Inhibitory transmission in locus coeruleus neurons expressing GABAA receptor epsilon subunit has a number of unique properties. , Belujon P., J Neurophysiol. October 1, 2009; 102 (4): 2312-25.
Pharmacological Properties of DOV 315,090, an ocinaplon metabolite. , Berezhnoy D., BMC Pharmacol. June 13, 2008; 8 11.
alpha1beta2delta, a silent GABAA receptor: recruitment by tracazolate and neurosteroids. , Zheleznova N., Br J Pharmacol. March 1, 2008; 153 (5): 1062-71.
Electrophysiological properties and subunit composition of GABAA receptors in patients with gelastic seizures and hypothalamic hamartoma. , Wu J ., J Neurophysiol. July 1, 2007; 98 (1): 5-15.
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities. , Hadley SH., J Physiol. June 15, 2007; 581 (Pt 3): 1001-18.
Changes in the function of the inhibitory neurotransmitter system in the rat brain following subchronic inhalation exposure to 1-bromopropane. , Ueno S ., Neurotoxicology. March 1, 2007; 28 (2): 415-20.
Interleukin-1beta enhances GABAA receptor cell-surface expression by a phosphatidylinositol 3-kinase/Akt pathway: relevance to sepsis-associated encephalopathy. , Serantes R., J Biol Chem. May 26, 2006; 281 (21): 14632-43.
Impact of epsilon and theta subunits on pharmacological properties of alpha3beta1 GABAA receptors expressed in Xenopus oocytes. , Ranna M., BMC Pharmacol. January 13, 2006; 6 1.
Selective GABAA alpha5 benzodiazepine inverse agonist antagonizes the neurobehavioral actions of alcohol. , Cook JB., Alcohol Clin Exp Res. August 1, 2005; 29 (8): 1390-401.
Abnormal GABAA receptors from the human epileptic hippocampal subiculum microtransplanted to Xenopus oocytes. , Palma E ., Proc Natl Acad Sci U S A. February 15, 2005; 102 (7): 2514-8.
Salicylidene salicylhydrazide, a selective inhibitor of beta 1-containing GABAA receptors. , Thompson SA., Br J Pharmacol. May 1, 2004; 142 (1): 97-106.
Characterization of wild-type (R100R) and mutated (Q100Q) GABAA alpha 6 subunit in Sardinian alcohol non-preferring rats (sNP). , Sanna A., Brain Res. March 28, 2003; 967 (1-2): 98-105.