???pagination.result.count???
11-trifluoromethyl-phenyldiazirinyl neurosteroid analogues: potent general anesthetics and photolabeling reagents for GABAA receptors. , Chen ZW., Psychopharmacology (Berl). September 1, 2014; 231 (17): 3479-91.
Relative positioning of classical benzodiazepines to the γ2-subunit of GABAA receptors. , Middendorp SJ., ACS Chem Biol. August 15, 2014; 9 (8): 1846-53.
Engineering a light-regulated GABAA receptor for optical control of neural inhibition. , Lin WC., ACS Chem Biol. July 18, 2014; 9 (7): 1414-9.
Modulation of ionotropic GABA receptors by 6-methoxyflavanone and 6-methoxyflavone. , Hall BJ., Neurochem Res. June 1, 2014; 39 (6): 1068-78.
Sh-I-048A, an in vitro non-selective super-agonist at the benzodiazepine site of GABAA receptors: the approximated activation of receptor subtypes may explain behavioral effects. , Obradović ALj., Dev Biol. March 20, 2014; 1554 36-48.
Neurosteroid analogues. 18. Structure-activity studies of ent-steroid potentiators of γ-aminobutyric acid type A receptors and comparison of their activities with those of alphaxalone and allopregnanolone. , Qian M., J Med Chem. January 9, 2014; 57 (1): 171-90.
GABAA receptors containing ρ1 subunits contribute to in vivo effects of ethanol in mice. , Blednov YA., PLoS One. January 1, 2014; 9 (1): e85525.
Fractalkine/CX3CL1 modulates GABAA currents in human temporal lobe epilepsy. , Roseti C., Epilepsia. October 1, 2013; 54 (10): 1834-44.
New insights in endogenous modulation of ligand-gated ion channels: histamine is an inverse agonist at strychnine sensitive glycine receptors. , Kletke O., Eur J Pharmacol. June 15, 2013; 710 (1-3): 59-66.
Subtype selectivity of α+β- site ligands of GABAA receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors. , Varagic Z., Br J Pharmacol. May 1, 2013; 169 (2): 384-99.
Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface. , Varagic Z., Br J Pharmacol. May 1, 2013; 169 (2): 371-83.
Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α1 GABA(A) receptors. , Joksimović S., Eur Neuropsychopharmacol. May 1, 2013; 23 (5): 390-9.
Additive inhibition of human α1β2γ2 GABAA receptors by mixtures of commonly used drugs of abuse. , Hondebrink L., Neurotoxicology. March 1, 2013; 35 23-9.
Macroscopic kinetics of pentameric ligand gated ion channels: comparisons between two prokaryotic channels and one eukaryotic channel. , Laha KT., PLoS One. January 1, 2013; 8 (11): e80322.
Structural link between γ-aminobutyric acid type A ( GABAA) receptor agonist binding site and inner β-sheet governs channel activation and allosteric drug modulation. , Venkatachalan SP., J Biol Chem. February 24, 2012; 287 (9): 6714-24.
The biochemical anatomy of cortical inhibitory synapses. , Heller EA., PLoS One. January 1, 2012; 7 (6): e39572.
Cloning and characterization of GABAA α subunits and GABAB subunits in Xenopus laevis during development. , Kaeser GE., Dev Dyn. April 1, 2011; 240 (4): 862-73.
Activation and potentiation of human GABAA receptors by non-dioxin-like PCBs depends on chlorination pattern. , Antunes Fernandes EC., Toxicol Sci. November 1, 2010; 118 (1): 183-90.
GABAergic circuits control stimulus-instructed receptive field development in the optic tectum. , Richards BA., Nat Neurosci. September 1, 2010; 13 (9): 1098-106.
Agonist function of the recombinant alpha 4 beta 3 delta GABAA receptor is dependent on the human and rat variants of the alpha 4-subunit. , Wang MD., Clin Exp Pharmacol Physiol. July 1, 2010; 37 (7): 662-9.
A synthetic 18-norsteroid distinguishes between two neuroactive steroid binding sites on GABAA receptors. , Evers AS., J Pharmacol Exp Ther. May 1, 2010; 333 (2): 404-13.
About a snail, a toad, and rodents: animal models for adaptation research. , Roubos EW ., Front Endocrinol (Lausanne). January 1, 2010; 1 4.
Inhibitory transmission in locus coeruleus neurons expressing GABAA receptor epsilon subunit has a number of unique properties. , Belujon P., J Neurophysiol. October 1, 2009; 102 (4): 2312-25.
Unanticipated structural and functional properties of delta-subunit-containing GABAA receptors. , Kaur KH., J Biol Chem. March 20, 2009; 284 (12): 7889-96.
Effect of dried bonito (katsuobushi) and some of its components on GABAA receptors. , Mitou M., Food Chem. June 1, 2008; 108 (3): 840-6.
Histamine action on vertebrate GABAA receptors: direct channel gating and potentiation of GABA responses. , Saras A., J Biol Chem. April 18, 2008; 283 (16): 10470-5.
alpha1beta2delta, a silent GABAA receptor: recruitment by tracazolate and neurosteroids. , Zheleznova N., Br J Pharmacol. March 1, 2008; 153 (5): 1062-71.
The antiepileptic drug levetiracetam stabilizes the human epileptic GABAA receptors upon repetitive activation. , Palma E ., Epilepsia. October 1, 2007; 48 (10): 1842-9.
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities. , Hadley SH., J Physiol. June 15, 2007; 581 (Pt 3): 1001-18.
Nootropic alpha7 nicotinic receptor allosteric modulator derived from GABAA receptor modulators. , Ng HJ., Proc Natl Acad Sci U S A. May 8, 2007; 104 (19): 8059-64.
Changes in the function of the inhibitory neurotransmitter system in the rat brain following subchronic inhalation exposure to 1-bromopropane. , Ueno S ., Neurotoxicology. March 1, 2007; 28 (2): 415-20.
Synthesis of trifluoromethylaryl diazirine and benzophenone derivatives of etomidate that are potent general anesthetics and effective photolabels for probing sites on ligand-gated ion channels. , Husain SS., J Med Chem. August 10, 2006; 49 (16): 4818-25.
Interleukin-1beta enhances GABAA receptor cell-surface expression by a phosphatidylinositol 3-kinase/Akt pathway: relevance to sepsis-associated encephalopathy. , Serantes R., J Biol Chem. May 26, 2006; 281 (21): 14632-43.
Pharmacological properties of GABAA receptors containing gamma1 subunits. , Khom S., Mol Pharmacol. February 1, 2006; 69 (2): 640-9.
Impact of epsilon and theta subunits on pharmacological properties of alpha3beta1 GABAA receptors expressed in Xenopus oocytes. , Ranna M., BMC Pharmacol. January 13, 2006; 6 1.
Stoichiometry and pharmacology of two human alpha4beta2 nicotinic receptor types. , Moroni M., J Mol Neurosci. January 1, 2006; 30 (1-2): 95-6.
Abnormal GABAA receptors from the human epileptic hippocampal subiculum microtransplanted to Xenopus oocytes. , Palma E ., Proc Natl Acad Sci U S A. February 15, 2005; 102 (7): 2514-8.
BDNF modulates GABAA receptors microtransplanted from the human epileptic brain to Xenopus oocytes. , Palma E ., Proc Natl Acad Sci U S A. February 1, 2005; 102 (5): 1667-72.
Fragrances in oolong tea that enhance the response of GABAA receptors. , Hossain SJ., Biosci Biotechnol Biochem. September 1, 2004; 68 (9): 1842-8.
Salicylidene salicylhydrazide, a selective inhibitor of beta 1-containing GABAA receptors. , Thompson SA., Br J Pharmacol. May 1, 2004; 142 (1): 97-106.
The interaction of anaesthetic steroids with recombinant glycine and GABAA receptors. , Weir CJ., Br J Anaesth. May 1, 2004; 92 (5): 704-11.
Flumazenil-independent positive modulation of gamma-aminobutyric acid action by 6-methylflavone at human recombinant alpha1beta2gamma2L and alpha1beta2 GABAA receptors. , Hall BJ., Eur J Pharmacol. April 26, 2004; 491 (1): 1-8.
Receptor subtype-dependent positive and negative modulation of GABA(A) receptor function by niflumic acid, a nonsteroidal anti-inflammatory drug. , Sinkkonen ST., Mol Pharmacol. September 1, 2003; 64 (3): 753-63.
The in vitro and in vivo enantioselectivity of etomidate implicates the GABAA receptor in general anaesthesia. , Belelli D., Neuropharmacology. July 1, 2003; 45 (1): 57-71.
Characterization of wild-type (R100R) and mutated (Q100Q) GABAA alpha 6 subunit in Sardinian alcohol non-preferring rats (sNP). , Sanna A., Brain Res. March 28, 2003; 967 (1-2): 98-105.
Neuronal representation of odourants in the olfactory bulb of Xenopus laevis tadpoles. , Czesnik D., Eur J Neurosci. January 1, 2003; 17 (1): 113-8.
Magnesium potentiation of the function of native and recombinant GABA(A) receptors. , Möykkynen T., Neuroreport. July 20, 2001; 12 (10): 2175-9.
Anesthetic properties of 4-iodopropofol: implications for mechanisms of anesthesia. , Lingamaneni R., Anesthesiology. June 1, 2001; 94 (6): 1050-7.
Effects of gaseous anesthetics nitrous oxide and xenon on ligand-gated ion channels. Comparison with isoflurane and ethanol. , Yamakura T., Anesthesiology. October 1, 2000; 93 (4): 1095-101.
Modulation by extracellular pH of GABAA receptors expressed in Xenopus oocytes injected with rat brain mRNA. , Robello M., Int J Neurosci. January 1, 2000; 103 (1-4): 41-51.